Aroylpiperidines and pyrrolidines. New class of potent central nervous system depressants Robert L. Duncan, Grover C. Helsley, William J. Welstead, John P. DaVanzo, William H. Funderburk, and Carl D. Lunsford pp 1 - 6; DOI: 10.1021/jm00295a001 |
Azabicyclo chemistry. I. Synthesis of 1,5-methano-7-methoxy-2,3,4,5-tetrahydro-1H-2-benzazepines. B-norbenzomorphans Arthur E. Jacobson and Michael Mokotoff pp 7 - 9; DOI: 10.1021/jm00295a002 |
3'-Methyl, 8-methyl, and 8-phenyl derivatives of 5,9-dimethyl-6,7-benzomorphans Albert Ziering, Nicholas Malatestinic, Thomas Williams, and Arnold Brossi pp 9 - 13; DOI: 10.1021/jm00295a003 |
Thioxanthene psychopharmacological agents. I. 9-(3-Aminopropyl)thioxanthene-2-sulfonamides James F. Muren and Barry M. Bloom pp 14 - 16; DOI: 10.1021/jm00295a004 |
Thioxanthene psychopharmacological agents. II. 9-(3-aminopropylidene)-N,N-dimethylthioxanthene-2-sulfonamides James F. Muren and Barry M. Bloom pp 17 - 23; DOI: 10.1021/jm00295a005 |
4'-Fluoro-4-(1,4,5,6-tetrahydroazepino[4,5-b]indol-3(2H)-yl)butyrophenones J. B. Hester, A. D. Rudzik, H. H. Keasling, and W. Veldkamp pp 23 - 26; DOI: 10.1021/jm00295a006 |
Analogs of .alpha.-methylphenethylamine (amphetamine). I. Synthesis and pharmacological activity of some methoxy and/or methyl analogs Beng-Thong Ho, William M. McIsaac, Rong An, L. Wayne Tansey, Kenneth E. Walker, Leo F. Englert, and Michael B. Noel pp 26 - 30; DOI: 10.1021/jm00295a007 |
Pharmacologic and metabolic studies with deuterated zoxazolamine Masato Tanabe, Josephine Tagg, Dennis Yasuda, Susanna E. LeValley, and Chozo Mitoma pp 30 - 32; DOI: 10.1021/jm00295a008 |
2-(4-Imidazolyl)cyclopropylamine Alfred Burger, Manuel Bernabe, and Paul Waddell Collins pp 33 - 35; DOI: 10.1021/jm00295a009 |
Novel type of substituted piperazine with high antiserotonin potency W. J. Van der Burg, I. L. Bonta, J. Delobelle, C. Ramon, and B. Vargaftig pp 35 - 39; DOI: 10.1021/jm00295a010 |
Effect of eight prostaglandins on platelet aggregation N. Chandra Sekhar pp 39 - 44; DOI: 10.1021/jm00295a011 |
Inhibition of viral neuraminidase by 1-phenoxymethyl-3,4-dihydroisoquinolines. I. Steric effects Michael S. Tute, Keith W. Brammer, Barry Kaye, and Reginald W. Broadbent pp 44 - 48; DOI: 10.1021/jm00295a012 |
Inhibition of viral neuraminidase by 1-phenoxymethyl-3,4-dihydroisoquinolines. II. Hansch analysis Michael S. Tute pp 48 - 51; DOI: 10.1021/jm00295a013 |
Metabolic fate of phenyltrimethylsilane and phenyldimethylsilane Ralph J. Fessenden and Ray A. Hartman pp 52 - 54; DOI: 10.1021/jm00295a014 |
Antifertility agents. IV. 2,3-Diphenylbenzo- and 5,6-polymethylenebenzofurans, 1,2-diphenylnaphthofurans, and some related compounds H. P. S. Chawla, P. K. Grover, Nitya Anand, V. P. Kamboj, and Amiya B. Kar pp 54 - 59; DOI: 10.1021/jm00295a015 |
Synthesis and hypoglycemic activity of substituted alkyl- and alkoxyguanidines Bernard J. Ludwig, David B. Reisner, Mervin Meyer, Leo S. Powell, Leon Simet, and Frank J. Stiefel pp 60 - 63; DOI: 10.1021/jm00295a016 |
Fluorinated pyrimidines. XXXIII. Synthesis of methylated 5-fluoro-2'-deoxyuridine derivatives Tasneem A. Khwaja and Charles Heidelberger pp 64 - 69; DOI: 10.1021/jm00295a017 |
Fluorinated pyrimidines. XXXIV. Structure-activity studies of methylated 5-fluoro-2'-deoxyuridine derivatives Raymond J. Kent, Tasneem A. Khwaja, and Charles Heidelberger pp 70 - 73; DOI: 10.1021/jm00295a018 |
Synthesis and thiolytic cleavage of S-acyl derivatives of 5-mercaptouracil and 5-mercapto-2'-deoxyuridine Michael P. Kotick, Thomas I. Kalman, and Thomas J. Bardos pp 74 - 77; DOI: 10.1021/jm00295a019 |
Cofactor inhibition of thymidylate synthetase. Tetrahydrofolic acid analogs Mathias P. Mertes and Ai Jeng Lin pp 77 - 82; DOI: 10.1021/jm00295a020 |
Irreversible enzyme inhibitors. CLXVI. Active-site-directed irreversible inhibitors of dihydrofolic reductase derived from 2,4-diamino-5-(3,4-dichlorophenyl)pyrimidine with 6 substituents and some factors in their cell wall transport Bernard Randall Baker and Nicolaas M. J. Vermeulen pp 82 - 86; DOI: 10.1021/jm00295a021 |
Irreversible enzyme inhibitors. CLXVII. Thymidine phosphorylase. 10. On the nature and dimensions of the hydrophobic bonding region. A Bernard Randall Baker and Stephen E. Hopkins pp 87 - 89; DOI: 10.1021/jm00295a022 |
6-Fluorotetracyclines Panayota Bitha, Joseph J. Hlavka, and James H. Boothe pp 89 - 92; DOI: 10.1021/jm00295a023 |
Predictability of correlations between in vitro tetracycline potencies and substituent indices Arthur Cammarata and Suh Jen Yau pp 93 - 97; DOI: 10.1021/jm00295a024 |
Antiprotozoal quinones. II. Synthesis of 4-amino-1,2-naphthoquinones and related compounds as potential antimalarials F. J. Bullock, J. F. Tweedie, D. D. McRitchie, and M. A. Tucker pp 97 - 103; DOI: 10.1021/jm00295a025 |
Synthetic schistosomicides. XIV. 1,4-Naphthoquinone mono(O-acyloximes), 4-amino-1,2-naphthoquinones, 2-amino-3-chloro-1,4-naphthoquinones, and other naphthoquinones Edward F. Elslager, Leslie M. Werbel, and Donald F. Worth pp 104 - 109; DOI: 10.1021/jm00295a026 |
Novel anthelmintic agents. IV. Noncyclic amidines related to pyrantel James W. McFarland and Harold L. Howes pp 109 - 113; DOI: 10.1021/jm00295a027 |
Novel anthelmintic agents. V. Thiazoline and dihydrothiazine analogs of pyrantel James W. McFarland, Harold L. Howes, L. H. Conover, J. E. Lynch, William C. Austin, and D. H. Morgan pp 113 - 119; DOI: 10.1021/jm00295a028 |
Quinoxaline studies. XV. Potential antimalarials. (RS)-.alpha.-(dialkylaminomethyl)-2-quinoxalinemethanols Henry R. Moreno and Harry Pershing Schultz pp 119 - 121; DOI: 10.1021/jm00295a029 |
Anthelmintic quaternary salts. V. 2-(p-Dialkylaminophenyl)-1-methylquinolinium salts G. Y. Paris, D. L. Garmaise, J. Komlossy, and R. C. McCrae pp 122 - 124; DOI: 10.1021/jm00295a030 |
Synthesis of .gamma.-dimethylamino-.alpha.-phenylcycloaklyl propionates as potential analgetics Mathias P. Mertes, Patrick E. Hanna, and Arthur A. Ramsey pp 125 - 128; DOI: 10.1021/jm00295a031 |
Insect chemosterilants. VIII. Boron compounds Joseph A. Settepani, Jerry B. Stokes, and Alexej B. Borkovec pp 128 - 131; DOI: 10.1021/jm00295a032 |
Optical isomers of metaraminol. Synthesis and biological activity Noel F. Albertson, F. C. McKay, H. E. Lape, J. O. Hoppe, W. H. Selberis, and A. Arnold pp 132 - 134; DOI: 10.1021/jm00295a033 |
Amphetamine analogs. II. Methylated phenethylamines Beng-Thong Ho, L. Wayne Tansey, Robert L. Balster, Rong An, William M. McIsaac, and Robert T. Harris pp 134 - 135; DOI: 10.1021/jm00295a034 |
Substituted quinazolonephenoxyethylhydrazines as monoamine oxidase inhibitors Surendra S. Parmar and Ramesh Chandra Arora pp 135 - 136; DOI: 10.1021/jm00295a035 |
Antiinflammatory agents. I. 3-Benzoylfluoroalkanesulfonanilides J. Kenneth Harrington, Jerry Earl Robertson, Donald C. Kvam, Robert R. Hamilton, Kelly T. McGurran, Ronald J. Trancik, Karl F. Swingle, George Gomer Innes Moore, and John F. Gerster pp 137 - 137; DOI: 10.1021/jm00295a036 |
1,4-Bis(2-indol-3-ylethyl)piperidines John L. Archibald, Thomas Baum, and Scott J. Childress pp 138 - 140; DOI: 10.1021/jm00295a037 |
Derivatives of 9-thioxanthenecarbonitrile James F. Muren pp 140 - 141; DOI: 10.1021/jm00295a038 |
Synthesis and hypoglycemic activity of 2-(.omega.-substituted alkylamino)-2-imidazolines D. B. Reisner, Bernard J. Ludwig, S. Gister, and K. Tomeczek pp 142 - 143; DOI: 10.1021/jm00295a039 |
Potential antidiabetics. Benzimidazole-2-sulfonylglycamide derivatives S. M. Deshpande, K. C. Datta, A. K. Sanyal, and M. K. Raina pp 143 - 144; DOI: 10.1021/jm00295a040 |
Conformational aspects of ureas in the inhibition of the Hill reaction Marvin R. Boots, Sharon G. Boots, and Donald E. Moreland pp 144 - 144; DOI: 10.1021/jm00295a041 |
1,2,3,4,6,7,12,12a-Octahydro-2-phenylpyrazino[2',1':6,1]pyrido[3,4-b]indole John W. Schulenberg and Donald F. Page pp 145 - 145; DOI: 10.1021/jm00295a042 |
Electronic factors in drug-receptor interactions Yvonne C. Martin pp 145 - 147; DOI: 10.1021/jm00295a043 |
.beta.-Amino ketones as inhibitors of pyruvic acid oxidation Rajendra S. Varma, Basheer Ali, Surendra S. Parmar, and W. Lewis Nobles pp 147 - 148; DOI: 10.1021/jm00295a044 |
Synthesis of 6-trifluoromethyl-1,4-dihydrazinophthalazine Bruno Cavalleri, Elvio Bellasio, and Anna Sardi pp 148 - 149; DOI: 10.1021/jm00295a045 |
Synthesis of the .alpha. and .beta. anomers of 1-(2-deoxy-D-ribofuranosyl)-2-pyridone Mathias P. Mertes pp 149 - 151; DOI: 10.1021/jm00295a046 |
Fluorinated pyrimidines. XXXVI. Synthesis of some 2,4-substituted 5-trifluoromethylpyrimidines Heino Diringer, Tasneem A. Khwaja, and Charles Heidelberger pp 151 - 152; DOI: 10.1021/jm00295a047 |
Synthesis and activity of a new class of heterocyclic compounds against Entamoeba histolytica. 1,2,3,3a-Tetrahydro-1-alkylcyclopenta[de]quinolines A. U. Dey and B. Pathak pp 152 - 153; DOI: 10.1021/jm00295a048 |
Antimalarials. 4-Substituted 1H-pyrazolo[3,4-b]quinolines Robert G. Stein, John H. Biel, and Tara Singh pp 153 - 155; DOI: 10.1021/jm00295a049 |
Febrifugine antimalarial agents. I. Pyridine analogs of febrifugine Morris Fishman and Philip A. Cruickshank pp 155 - 156; DOI: 10.1021/jm00295a050 |
Synthesis and antimalarial activity of amodiaquine analogs Ned D. Heindel and James Molnar pp 156 - 157; DOI: 10.1021/jm00295a051 |
Arylglyoxal N,N-disubstituted hydrazones with antiviral and antifungal activity Elena Massarani, Dante Nardi, R. Pozzi, and L. Degen pp 157 - 159; DOI: 10.1021/jm00295a052 |
Synthesis and antimicrobial activity of some thenoyl amides M. Likar, P. Schauer, M. Japelj, M. Globokar, M. Oklobdzija, A. Povse, and V. Sunjic pp 159 - 161; DOI: 10.1021/jm00295a053 |
Synthesis of 5,8-quinazolinedione Giorgio Malesani, Francesco Marcolin, and Giovanni Rodighiero pp 161 - 162; DOI: 10.1021/jm00295a054 |
Terpene compounds as drugs. VII. Terpenylhydroxamic acids Silvano Casadio, Antonio Mantegani, Amedeo Omodei Sale, and Germano Coppi pp 162 - 164; DOI: 10.1021/jm00295a055 |
Nitrofuryl heterocycles. IX. Some derivatives and analogs of 6,7-dihydro-3-(5-nitro-2-furyl)-5H-imidazo[2,1-b]thiazolium chloride Harry R. Snyder and Louis E. Benjamin pp 164 - 165; DOI: 10.1021/jm00295a056 |
Diethylaminoethyl ethers of coumarins Satyendra Kumar pp 166 - 166; DOI: 10.1021/jm00295a057 |
Reaction of chloroquinolines with formamides Ned D. Heindel and Peter D. Kennewell pp 166 - 167; DOI: 10.1021/jm00295a058 |
Synthesis of 3-bromo- and 3-chloro-1-methyl-4-phenyl-4-propionoxypiperidines as potential analgetics Philip M. Carabateas pp 167 - 167; DOI: 10.1021/jm00295a059 |
The American Society for Pharmacology and Experimental Therapeutics. The First Sixty Years. 1908-1969 Alfred Burger pp 168 - 168; DOI: 10.1021/jm00295a900 |
Solid Phase Peptide Synthesis Keith O. Hodgson pp 168 - 168; DOI: 10.1021/jm00295a901 |
Annual Reports in Medicinal Chemistry, 1968. Alfred Burger pp 168 - 168; DOI: 10.1021/jm00295a902 |
.beta.-Adrenergic blocking agents. VII. 2-(1,4-Benzodioxanyl) and 2-chromanyl analogs of pronethalol [2-isopropylamino-1-(2-naphthyl) ethanol] Ralph Howe, Balbir S. Rao, and M. S. Chodnekar pp 169 - 176; DOI: 10.1021/jm00296a001 |
Analogs of angiotensin II. I. Solid phase synthesis N. C. Chaturvedi, Won Kil Park, R. R. Smeby, and F. M. Bumpus pp 177 - 181; DOI: 10.1021/jm00296a002 |
Analogs of angiotensin II. II. Mechanism of receptor interaction Philip A. Khairallah, A. Toth, and F. M. Bumpus pp 181 - 184; DOI: 10.1021/jm00296a003 |
[2,4-Diisoleucine]-oxytocin. Analog of oxytocin with natriuretic and diuretic activities Victor J. Hruby, Vincent Du Vigneaud, and Wah-Yip Chan pp 185 - 187; DOI: 10.1021/jm00296a004 |
Pyridoxine chemistry. XXII. Selective modifications of the .alpha.4-position of pyridoxol. I. Extension and branching of the 4-side chain Wsewolod Korytnyk and Burton Paul pp 187 - 191; DOI: 10.1021/jm00296a005 |
Antidepressants. II. Bridged ring ether derivatives in the dibenzocycloheptene series Marcia E. Christy, Carole C. Boland, June G. Williams, and Edward L. Engelhardt pp 191 - 195; DOI: 10.1021/jm00296a006 |
Synthesis and activity of some 3-substituted 1,2,3,4-pseudooxatriazol-5-ones and their precursors and related compounds T. L. Thomas, M. Fedorchuk, B. V. Shetty, and F. E. Anderson pp 196 - 203; DOI: 10.1021/jm00296a007 |
Nonsteroidal antiinflammatory agents. I. 6-Substituted 2-naphthylacetic acids Ian Thomas Harrison, Brian Lewis, Peter Nelson, Wendell Rooks, Adolph Roszkowski, Albert Tomolonis, and John H. Fried pp 203 - 205; DOI: 10.1021/jm00296a008 |
Preparation and antiinflammatory activity of some 2-arylbenzo[b] thiophen-3(2H)-one 1,1-dioxides Joseph G. Lombardino and Edward H. Wiseman pp 206 - 210; DOI: 10.1021/jm00296a009 |
Synthesis and pharmacological properties of substituted cinnamohydroxamic acids N. P. Buu-Hoi, Claude L. Gillet, Georges E. Lambelin, Jose L. Roba, and Jacques E. Thiriaux pp 211 - 213; DOI: 10.1021/jm00296a010 |
Sulfur and selenium compounds related to acetylcholine and choline. X. Acetylthionocholine Shih-Hsi Chu and Henry G. Mautner pp 214 - 215; DOI: 10.1021/jm00296a011 |
In vitro inhibition of cholesterolgenesis by various thyroid hormone analogs Cleamond D. Eskelson, Clarence R. Cazee, W. Anthony, Jack C. Towne, and Benedict R. Walske pp 215 - 220; DOI: 10.1021/jm00296a012 |
Choline acetyltransferase inhibitors. Dimensional and substituent effects among styrylpyridine analogs Chester J. Cavallito, H. S. Yun, T. Kaplan, John Crispin Smith, and Francis F. Foldes pp 221 - 224; DOI: 10.1021/jm00296a013 |
Structure-activity relations. I. Series of antagonists of acetylcholine and histamine at the postganglionic receptors Keith Bowden and Rodney Christopher Young pp 225 - 230; DOI: 10.1021/jm00296a014 |
Antimalarials. 8-chloro-4-(2'-N,N-dibutylamino-1'-hydroxyethyl) benzo[h]-1,6-naphthyridine Karl A. Roseman, Maribeth M. Gould, Warner M. Linfield, and Ben E. Edwards pp 230 - 233; DOI: 10.1021/jm00296a015 |
Syntheses of phenanthrene amino alcohols as antimalarials Leroy Krbechek, Richard R. Riter, Richard G. Wagner, and Clarence W. Huffman pp 234 - 238; DOI: 10.1021/jm00296a016 |
Nitrones. II. .alpha.-(5-Nitro-2-furyl)-N-cycloalkyl- and -N-alkylnitrones Hyun Koo Kim, Hesham K. Yaktin, and Ronald E. Bambury pp 238 - 241; DOI: 10.1021/jm00296a017 |
N-sulfanilyl-l-alkylcytosines. New highly active class of "soluble," short-acting sulfanilamides Leonard Doub, Uldis Krolls, J. M. Vandenbelt, and Myron W. Fisher pp 242 - 246; DOI: 10.1021/jm00296a018 |
Preparation and antibacterial activity of some sulfanilamidodiazines bearing the N-alkylalkanesulfonamido group William E. Kreighbaum, Frederick A. Grunwald, Edward F. Harrison, John A. LaBudde, and A. A. Larsen pp 247 - 251; DOI: 10.1021/jm00296a019 |
Potential antiradiation agents. III. N-substituted aminoethane-thiosulfuric acids Daniel L. Klayman, Marie M. Grenan, and David P. Jacobus pp 251 - 254; DOI: 10.1021/jm00296a020 |
Antiviral agents. I. Bicyclo[2.2.2]octan- and -oct-2-enamines Joel G. Whitney, W. A. Gregory, J. C. Kauer, J. R. Roland, Jack A. Snyder, R. E. Benson, and E. C. Hermann pp 254 - 260; DOI: 10.1021/jm00296a021 |
Antiprotozoal quinones. III. Synthesis of 8-amino-5,6-quinolinediones, 8-amino-7-chloro-5,6-quinolinediones, and 8-amino-5,5,7-trichloro-6(5H)-quinolones as potential antimalarials F. J. Bullock and J. F. Tweedie pp 261 - 264; DOI: 10.1021/jm00296a022 |
Preparation and the results of antitumor screening of some substituted amino-, azido-, halogeno- and hydroxy-p-benzoquinones Kwang-Yuen Zee-Cheng and Chia-Chung Cheng pp 264 - 268; DOI: 10.1021/jm00296a023 |
Nucleosides. LXIV. Fluoro sugar analogs of arabinosyl- and xylosylcytosines John Arthur Wright, Dan Patrick Wilson, and Jack J. Fox pp 269 - 272; DOI: 10.1021/jm00296a024 |
Effect of some heterocyclic disulfides and thiones on the carbohydrate metabolism of Ehrlich ascites tumor Davide R. Grassetti, John F. Murray, M. E. Brokke, and A. D. Gutman pp 273 - 276; DOI: 10.1021/jm00296a025 |
Cofactor inhibitors of thymidylate synthetase. Piperidine and tetrahydroquinoline analogs of tetrahydrofolic acid Mathias P. Mertes and Ai Jeng Lin pp 276 - 279; DOI: 10.1021/jm00296a026 |
Irreversible enzyme inhibitors. CLXVIII. Irreversible inhibition of dihydrofolate reductase and cell wall transport by pyrimidines and dihydro-s-triazines with pyridinium side chains Bernard Randall Baker, Nicolaas M. J. Vermeulen, and Adrian J. Ryan pp 280 - 284; DOI: 10.1021/jm00296a027 |
Mixed bifunctionality. II. Relation of antitumor activity to structure in alkylating agents derived from polynuclear aromatic hydrocarbons Richard M. Peck, Anna P. O'Connell, and Hugh J. Creech pp 284 - 288; DOI: 10.1021/jm00296a028 |
Nitrofuryl heterocycles. X. Analogs of 6-(5-nitro-2-furyl)-as-triazine-3,5(2H,4H)-dione Homer A. Burch pp 288 - 291; DOI: 10.1021/jm00296a029 |
Nitrofuryl heterocycles. XI. 3-(5-Nitro-2-furyl)-.DELTA.2-1,2,4-triazolin-5-ones Louis E. Benjamin, Homer A. Burch, and Richard Dobson pp 291 - 292; DOI: 10.1021/jm00296a030 |
Synthesis of 1-phenyl-2-styryl-3,5-dioxopyrazolidines as antiinflammatory agents Hisao Yamamoto and Shinichi Kaneko pp 292 - 295; DOI: 10.1021/jm00296a031 |
2-Trifluoromethoxydibenz[b,e][1,4]diazepine and 2-trifluoromethoxydibenz[b,f][1,4]-oxazepine derivatives Francis J. McEvoy, E. N. Greenblatt, A. C. Osterberg, and George Rodger Allen pp 295 - 297; DOI: 10.1021/jm00296a032 |
.alpha.,.alpha.,.alpha.-Trifluorotoluic acid (5-nitrofurfurylidene)hydrazides Dean E. Welch, Harry S. Nakaue, and Robert D. Vatne pp 297 - 298; DOI: 10.1021/jm00296a033 |
Comparison of some stereochemical requirements of the acetyl-cholinesterase and muscarinic receptor areas George H. Cocolas, Ellen Chenault Robinson, and William L. Dewey pp 299 - 301; DOI: 10.1021/jm00296a034 |
Phosphorus-nitrogen compounds. XI. Phosphamidase studies. I. Unsubstituted amides Lindley A. Cates pp 301 - 302; DOI: 10.1021/jm00296a035 |
Synthesis of pentazocine Noel F. Albertson and William F. Wetterau pp 302 - 303; DOI: 10.1021/jm00296a036 |
Substituted benzamides. Analogs of .beta.-hydroxyethylcyclohexylamine with CNS [central nervous system] depressant and hypotensive activity William D. Roll pp 303 - 304; DOI: 10.1021/jm00296a037 |
Synthesis of some local anesthetics Pramod K. Srivastava and P. N. Srivastava pp 304 - 305; DOI: 10.1021/jm00296a038 |
Synthesis of compounds with potential central nervous system stimulant activity. II. 5-Spiro-substituted 2-amino-2-oxazolines Michael R. Harnden and Ray R. Rasmussen pp 305 - 308; DOI: 10.1021/jm00296a039 |
3-Substituted 1,2,3,4-tetrahydrocarbazoles Leonard M. Rice and Kenneth Richard Scott pp 308 - 311; DOI: 10.1021/jm00296a040 |
16-Oxygenated 17.alpha.-methyl-5.beta.-androstanes Tadashi Watabe, Sachiko Yagishita, and Shoji Hara pp 311 - 312; DOI: 10.1021/jm00296a041 |
Synthesis of 1-(3'-N,N-diethylaminopropyl)-2-alkylnaphth[1,2-d]-imidazole-4,5-diones F. Ivy Carroll, J. T. Blackwell, and H. Wayne Miller pp 312 - 314; DOI: 10.1021/jm00296a042 |
Analogs of steroid hormones. III. Benz[e]indene derivatives Richard E. Juday, Bonnie Bukwa, Kent Kaiser, and Gordon Webb pp 314 - 317; DOI: 10.1021/jm00296a043 |
Organic disulfides and related substances. XXVIII. Analogs of o-(2-protoaminoethyldithio)benzoate as antiradiation drugs Lamar Field and Patton M. Giles pp 317 - 319; DOI: 10.1021/jm00296a044 |
Effect of organic compounds on reproductive processes. VIII. Methanesulfonyloxyacetyl derivatives of diamines Wilfred A. Skinner and J. G. Johansson pp 319 - 320; DOI: 10.1021/jm00296a045 |
Cassaine analogs. VI. Resolution of (.dag.)-7-deoxy-16,17,18,20-tetranorcassaic acid and biological activity of derived esters Robert LaGrone Clarke and Sol J. Daum pp 320 - 322; DOI: 10.1021/jm00296a046 |
Preparation and fungistatic properties of thiocarbohydrazones David M. Wiles and Tony Suprunchuk pp 323 - 324; DOI: 10.1021/jm00296a047 |
Antiprotozoal 4-aryloxy-2-aminoquinolines and related compounds Diether G. Markees, Virginia C. Dewey, and George W. Kidder pp 324 - 326; DOI: 10.1021/jm00296a048 |
Antimalarials. 4,4'-Diaminodiphenyl sulfone-type compounds Tara Singh, Robert George Stein, and John H. Biel pp 326 - 327; DOI: 10.1021/jm00296a049 |
Synthetic trypanocides. I. Substituted 1,2,3,4-tetrahydrocarbazoles Jorge G. Pecca and Sem M. Albonico pp 327 - 328; DOI: 10.1021/jm00296a050 |
Derivatives of 2-hydroxy-p-phenetidine. I. Azomethines Moses J. Namkung and T. Lloyd Fletcher pp 329 - 329; DOI: 10.1021/jm00296a051 |
2,3-Dihydro-4(1H)-quinazolinone derivatives Giuseppe Bonola and Enrico Sianesi pp 329 - 332; DOI: 10.1021/jm00296a052 |
Hexachlorocyclopentadiene adducts of unsaturated amides Robert R. Mod, Frank C. Magne, Evald L. Skau, and Gene Sumrell pp 332 - 333; DOI: 10.1021/jm00296a053 |
4-Demethyltrichocereine Sidney Teitel and Arnold Brossi pp 333 - 333; DOI: 10.1021/jm00296a054 |
Quaternization products of S-(--)-nicotine Charles H. Jarboe and Charlotte M. Schmidt pp 333 - 334; DOI: 10.1021/jm00296a055 |
1-Arylsulfonylhydrazides. III. 4-Phenyl-1-arylsulfonylthiosemicarbazides and 2-arylsulfonylhydrazone-3-phenyl-4-thiazolines Carlos Sunkel and Humberto Gomez pp 334 - 335; DOI: 10.1021/jm00296a056 |
Aminopyrimidine steroid David M. Piatak and Eliahu Caspi pp 335 - 335; DOI: 10.1021/jm00296a057 |
Antituberculous Schiff bases Jaysukhlal R. Merchant and D. S. Chothia pp 335 - 336; DOI: 10.1021/jm00296a058 |
Principles of Drug Action. The Basis of Pharmacology Avram Goldstein, Lewis Aronow, and Sumner M. Kalman pp 337 - 337; DOI: 10.1021/jm00296a900 |
Circulatory Drugs. Pharmacological and Clinical Approach to the Detection and Evaluation of New Circulatory Drugs A. Bertelli pp 337 - 337; DOI: 10.1021/jm00296a901 |
Pharmaceutical Chemistry. Part II: Inorganic M.L. Schroff pp 337 - 337; DOI: 10.1021/jm00296a902 |
Atlas of Protein Sequence and Structure 1969 Alfred Burger pp 337 - 337; DOI: 10.1021/jm00296a903 |
Isolation and Identification of Drugs in Pharmaceuticals. Body Fluids, and Post-mortem Material pp 338 - 338; DOI: 10.1021/jm00296a905 |
Polypeptides. XLV. Structure-function studies in the .beta.-corticotropin series Klaus Hofmann, Rudolf Andreatta, Hans Bohn, and Luis Moroder pp 339 - 345; DOI: 10.1021/jm00297a001 |
Synthesis and pharmacological properties of 4-decarboxamido-8-arginine-vasopressin and its 1-deamino analog Dieter Gillessen and Vincent Du Vigneaud pp 346 - 349; DOI: 10.1021/jm00297a002 |
Synthesis of analogs of the C-terminal octapeptide of cholecystokinin-pancreozymin. Structure-activity relation Josip Pluscec, John T. Sheehan, Emily F. Sabo, Nina Williams, Octavian Kocy, and Miguel A. Ondetti pp 349 - 352; DOI: 10.1021/jm00297a003 |
Angiotensin II analogs. III. Synthesis and biological evaluation of some des-aspartyl-angiotensins Eugene C. Jorgensen, Graham C. Windridge, and Thomas Choy Lee pp 352 - 356; DOI: 10.1021/jm00297a004 |
Synthesis and positive inotropic effect of strophanthidol 3-bromoacetate-19-3H Richard Edward Thomas, Barbara F. Roth-Schechter, and George T. Okita pp 357 - 359; DOI: 10.1021/jm00297a005 |
Hypocholesteremic agents. I. Substituted stilbazoles and dihydrostilbazoles Frank J. Villani, Claire A. Ellis, Robert F. Tavares, Merl Steinberg, and Sibylle Tolksdorf pp 359 - 366; DOI: 10.1021/jm00297a006 |
Thyroxine analogs. XVIII. 3,5-Dialkyl-3'-halo-DL-thyronines and their 3'-methyl and 4'-amino analogs Eugene C. Jorgensen and Jeremy Wright pp 367 - 370; DOI: 10.1021/jm00297a007 |
Synthetic schistosomicides. XVI. 5-(Mono- and dialkylamino)-2-nitrosophenols, 2-amino-5-(dialkylamino)phenols, and related compounds Edward F. Elslager and Donald F. Worth pp 370 - 376; DOI: 10.1021/jm00297a008 |
N-substituted N'-hydroxythioureas Gil Clifton, Sarah R. Bryant, and Charles G. Skinner pp 377 - 379; DOI: 10.1021/jm00297a009 |
8-Hydroxyquinoline derivatives. Synthesis and biological evaluation of arylglyoxal N-7-amino-5-substituted 8-hydroxyquinoline hemiacetals and 5-phenylglyoxylidenamino-8-hydroxyquinolines Elena Massarani, Dante Nardi, R. Pozzi, L. Degen, and Maria J. Magistretti pp 380 - 383; DOI: 10.1021/jm00297a010 |
Potential antimalarials. IV. Quinoline-.alpha.,.alpha.-dialkylmethanols Joel B. Wommack and Donald E. Pearson pp 383 - 386; DOI: 10.1021/jm00297a011 |
Chemical conversion of desacetylcephalothin lactone into desacetylcephalothin. The final link in a total synthesis of cephalosporanic acid derivatives Saul L. Neidleman, Samuel C. Pan, Jerold A. Last, and Joseph E. Dolfini pp 386 - 388; DOI: 10.1021/jm00297a012 |
Transformations of 6-phenylacetamido- and 6-tritylaminopenicillanyl p-toluenesulfonate and p-nitrobenzenesulfonate Malcolm Rice Bell, Stephen D. Clemans, and Rudolf Oesterlin pp 389 - 394; DOI: 10.1021/jm00297a013 |
2-Tetrahydropyridylindoles as histamine and serotonin antagonists Robert N. Schut, Frederick E. Ward, O. J. Lorenzetti, and Enrique Hong pp 394 - 397; DOI: 10.1021/jm00297a014 |
.beta.-Adrenergic blocking agents. VIII. Reactions of .beta.-haloalkylamines related to pronethalol and propranolol Ralph Howe pp 398 - 403; DOI: 10.1021/jm00297a015 |
New class of sympathetic .beta.-receptor blocking agents. 3,4-Dihydro-3-hydroxy-1,5-benzoxazocines Berkeley Basil, E. C. J. Coffee, D. L. Gell, Donald R. Maxwell, D. J. Sheffield, and Kenneth R. H. Wooldridge pp 403 - 406; DOI: 10.1021/jm00297a016 |
Synthesis of 6-(N-alkyl-N-arylamino)pyrimidines as potential antimetabolites Paul L. Warner and Thomas J. Bardos pp 407 - 410; DOI: 10.1021/jm00297a017 |
Preparation and activity of the 4'-thio-derivatives of some 6-substituted purines nucleosides Miroslav Bobek, Roy L. Whistler, and Alexander Bloch pp 411 - 413; DOI: 10.1021/jm00297a018 |
Experimental antileukemic agents. Preparation and structure-activity study of S-tritylcysteine and related compounds Kwang-Yuen Zee-Cheng and Chia-Chung Cheng pp 414 - 418; DOI: 10.1021/jm00297a019 |
Synthesis and pharmacological evaluation of .alpha.-naphthylalkylamines Silvano Casadio, Gianfranco Pala, Tiberio Bruzzese, Carla Turba, and Ernesta Marazzi-Uberti pp 418 - 421; DOI: 10.1021/jm00297a020 |
Anticancer agents. IV. Antitumor activity of some 1,4- and 1,5-(bisthiosemicarbazones) and of related heterocycles Vincent C. Barry, Michael L. Conalty, Joan E. McCormick, Robert S. McElhinney, Mary R. McInerney, and John F. O'Sullivan pp 421 - 427; DOI: 10.1021/jm00297a021 |
2-Fluoropurine ribonucleosides John A. Montgomery and Kathleen Hewson pp 427 - 430; DOI: 10.1021/jm00297a022 |
Potential antitumor agents. IV. 4-Substituted 1-formylisoquinoline thiosemicarbazones Krishna C. Agrawal, Robert J. Cushley, Walter J. McMurray, and Alan C. Sartorelli pp 431 - 434; DOI: 10.1021/jm00297a023 |
Model studies for the reactivation of aged phosphonylated acetylcholinesterase. Use of alkylating agents containing nucleophilic groups George M. Steinberg, Claire N. Lieske, Roger Boldt, John C. Goan, and Harold E. Podall pp 435 - 446; DOI: 10.1021/jm00297a024 |
Alkylating agents related to 2,2'-biaziridine. III. Stereoisomeric N,N'-dimethylsulfonyl-2,2'-biaziridines Peter W. Feit and Ole T. Nielsen pp 447 - 452; DOI: 10.1021/jm00297a025 |
Structure-activity relations in adenosine deaminase inhibitors Howard J. Schaeffer, Roland Norman Johnson, E. Odin, and Corwin Hansch pp 452 - 455; DOI: 10.1021/jm00297a026 |
Irreversible enzyme inhibitors. CLXIX. Inhibition of FUDR [5-fluoro-2'-deoxyuridine] phosphorylase from Walker 256 rat tumor by 6-substituted uracils Bernard Randall Baker and James L. Kelley pp 456 - 458; DOI: 10.1021/jm00297a027 |
Irreversible enzyme inhibitors. CLXX. Inhibition of FUDR [5-fluoro-2'-deoxyuridine] phosphorylase from Walker 256 rat tumor by 1-substituted uracils Bernard Randall Baker and James L. Kelley pp 458 - 461; DOI: 10.1021/jm00297a028 |
Irreversible enzyme inhibitors. CLXXI. Inhibition of FUDR [5-fluoro-2'-deoxyuridine] phosphorylase from Walker 256 rat tumor by 5-substituted uracils Bernard Randall Baker and James L. Kelley pp 461 - 467; DOI: 10.1021/jm00297a029 |
Irreversible enzyme inhibitors. CLXXII. Proteolytic enzymes. XVI. Covalent bonding of the sulfonyl fluoride group to serine outside the active-site of .alpha.-chymotrypsin by exo-type active-site directed irreversible inhibitors Robert Cardinaud and Bernard Randall Baker pp 467 - 470; DOI: 10.1021/jm00297a030 |
Nucleophilicity of heteroaromatic aldoximes bearing an aminoalkyl side chain. IV Yacov Ashani and Sasson Cohen pp 471 - 474; DOI: 10.1021/jm00297a031 |
Mechanism of metabolic 3-hydroxylation of benzodiazepines. Fragmentation pattern of 1,4-benzodiazepin-2-ones under electron impact Wolfgang Sadee pp 475 - 479; DOI: 10.1021/jm00297a032 |
Agents acting on the central nervous system. XII. 3-Tert-aminopropiophenones as central muscle relaxants and diuretics H. P. S. Chawla, B. C. Gautam, R. S. Kapil, Nitya Anand, G. K. Patnaik, Man M. Vohra, and O. P. Shrivastava pp 480 - 488; DOI: 10.1021/jm00297a033 |
1,2,3,4,5,6-Hexahydro-6-phenyl-2,6-methano-3-benzazocines. II Naokata Yokoyama, Fred B. Block, and Frank H. Clarke pp 488 - 492; DOI: 10.1021/jm00297a034 |
Linear free energy relations in the alkaline hydrolysis of substituted benzoylcholine esters James J. Zimmerman and Jere E. Goyan pp 492 - 497; DOI: 10.1021/jm00297a035 |
Metabolism of pyrovalerone hydrochloride Werner Michaelis, Jeff H. Russel, and Othmar Schindler pp 497 - 503; DOI: 10.1021/jm00297a036 |
Structure-dependent inhibition by synthetic fibrinolytic anions of collagen-induced aggregation of human platelets Detlev Thilo and Kurt N. Von Kaulla pp 503 - 510; DOI: 10.1021/jm00297a037 |
Influence of lipophilic character on the antibacterial activity of cephalosporins and penicillins Gian L. Biagi, Maria C. Guerra, Anna M. Barbaro, and Maria F. Gamba pp 511 - 516; DOI: 10.1021/jm00297a038 |
Agents acting on the central nervous system. XIII. 2,3,4,4a,5,6-Hexahydro-1(H)-pyrazino[1,2-a]quinolines. A new class of hypotensive agents V. Aruna Rao, Padam C. Jain, Nitya Anand, R. C. Srimal, and Prithvi R. Dua pp 516 - 522; DOI: 10.1021/jm00297a039 |
Benzo[g]quinolines. II. Novel synthesis and pharmacological evaluation of cis-1-alkyl-1,2,3,4,4a,5,10,10a-octahydrobenzo[g]quinolines William F. Michne and Noel F. Albertson pp 522 - 525; DOI: 10.1021/jm00297a040 |
Novel analgetics and molecular rearrangements in the morphine-thebaine group. XVIII. 3-Deoxy-6,14-endo-etheno-6,7,8,14-tetrahydrooripavines John William Lewis and Michael J. Readhead pp 525 - 527; DOI: 10.1021/jm00297a041 |
Central nervous system stimulants of the xanthone series Paolo Da Re, Laura Sagramora, Vittorio Mancini, P. Valenti, and Lorenzo Cima pp 527 - 531; DOI: 10.1021/jm00297a042 |
Thia steroids. III. Derivatives of 2-thia-A-nor-5.alpha.-androstan-17.beta.-ol as probes of steroid-receptor interactions Manfred E. Wolff, Galal Zanati, G. Shanmugasundarum, Sharad Gupte, and Gunhild Aadahl pp 531 - 534; DOI: 10.1021/jm00297a043 |
Potential naphthoquinone antimalarials. 2-Acylhydrazino-1,4-naphthoquinonones Kenneth H. Dudley and H. Wayne Miller pp 535 - 537; DOI: 10.1021/jm00297a044 |
Antimalarials. II. Quinolinemethanols with decreased phototoxicity Edward R. Atkinson and Anthony J. Puttick pp 537 - 541; DOI: 10.1021/jm00297a045 |
Antimalarials. Quinolinemethanol derivatives Tara Singh and John H. Biel pp 541 - 541; DOI: 10.1021/jm00297a046 |
Antimalarial substances. XXII. Synthetic schistosomicides. XV. Antimalarial and antischistosomal effects of .alpha.,.alpha.,.alpha.,.alpha.',.alpha.',.alpha.'-hexachloroxylene derivatives and related halogenated hydrocarbons Edward F. Elslager, Marland P. Hutt, and Leslie M. Werbel pp 542 - 544; DOI: 10.1021/jm00297a047 |
Coumarin derivatives as coronary vasodilators Dilbagh S. Bariana pp 544 - 546; DOI: 10.1021/jm00297a048 |
Antimalarials. Antagonists of pantothenic acid Raj K. Razdan, Catherine M. Reinsel, and Barbara A. Zitko pp 546 - 549; DOI: 10.1021/jm00297a049 |
Synthesis and microbiological properties of some substituted derivatives of 3-amino-3,4-dihydrocarbostyril Alvie L. Davis, James W. Hughes, Robert L. Hance, Vicki L. Gault, and Tommy J. McCord pp 549 - 550; DOI: 10.1021/jm00297a050 |
Antiprotozoal quinones. IV. 2-Amino-1,4-naphthoquinone imines as potential antimalarials Frank J. Bullock, John F. Tweedie, Donna D. McRitchie, and Margaret A. Tucker pp 550 - 552; DOI: 10.1021/jm00297a051 |
Substituted N-phenylanthranilic acid hydrazides as potential antimalarial and antimicrobial agents N. H. Berner, Rajendra S. Varma, and David W. Boykin pp 552 - 554; DOI: 10.1021/jm00297a052 |
1-Adamantanecarboxylic acid amide of 4-aminoantipyrine Remo Spano, G. Linari, and R. Marri pp 554 - 554; DOI: 10.1021/jm00297a053 |
2-(Substituted amino)quinolizinium bromides. A new class of anthelmintic agents Robert J. Alaimo, Christopher J. Hatton, and Michael K. Eckman pp 554 - 556; DOI: 10.1021/jm00297a054 |
Hypoglycemic activity of 1-alkenyl- and 1-alkenoyl-3-arylsulfonylureas Gianfranco Pala, Antonio Mantegani, Amedeo Omodei-Sale, and Germano Coppi pp 556 - 557; DOI: 10.1021/jm00297a055 |
New class of ultralong-acting local anesthetics James F. Stubbins, Seymour Ehrenpreis, T. H. Lynes, and M. Bigo-Gullino pp 558 - 559; DOI: 10.1021/jm00297a056 |
Radioopaque contrast media. XVIII. Derivatives of 2-(3-amino-2,4,6-triiodophenyl)alkanoic acids Ernst Felder, Davide Pitre, Luciano Fumagalli, and Enrico Lorenzotti pp 559 - 561; DOI: 10.1021/jm00297a057 |
Chlorosulfonation of 17.beta.-acetoxy-3-methoxyestra-1,3,5(10)-triene Arthur H. Goldkamp pp 561 - 563; DOI: 10.1021/jm00297a058 |
Thia steroids. II. 2-Thia-A-nor-5.alpha.-pregnan-20-one Manfred E. Wolff and Galal Zanati pp 563 - 563; DOI: 10.1021/jm00297a059 |
Pyrolysis of 16-methylene 17-oxygenated-20-keto steroids. IV. Synthesis of 3-hydroxy-1,3,5(10)-estratrienol[17,16-c]-2'-methylfuran Thomas L. Popper, Olga Gnoj, F. E. Carlon, and Merl Steinberg pp 564 - 565; DOI: 10.1021/jm00297a060 |
N-substituted 2,2'-diphenamic acids and diphenimides. I Carol A. Cole, Hsi-Lung Pan, Moses J. Namkung, and T. Lloyd Fletcher pp 565 - 567; DOI: 10.1021/jm00297a061 |
Derivatives of fluorene. XXXII. Diphenimides. 2. Some ring substituted N-2-fluorenyl-2',2"-diphenamic acids and diphenimides Hsi-Lung Pan and T. Lloyd Fletcher pp 567 - 568; DOI: 10.1021/jm00297a062 |
Synthesis of potential anticancer agents. 5,12-Naphthacene-quinones Jacob Finkelstein and John A. Romano pp 568 - 570; DOI: 10.1021/jm00297a063 |
Reduction of 1-(4-dimethylaminobenzylidene)indene Carl T. Bahner, David H. Brotherton, Thomas Harmon, and B. L. Stump pp 570 - 571; DOI: 10.1021/jm00297a064 |
Synthesis of additional arylhydroxamic acids which inhibit nucleic acid biosynthesis in vitro Glen R. Gale, John B. Hynes, and Alayne B. Smith pp 571 - 574; DOI: 10.1021/jm00297a065 |
Glycylureas and quaternary salts Price Truitt and J. T. Witkowski pp 574 - 574; DOI: 10.1021/jm00297a066 |
Antitumor activity of some azine and hydrazone derivatives of 1,4-dimethoxy-2-butanone William J. Haggerty and Chia-Chung Cheng pp 574 - 575; DOI: 10.1021/jm00297a067 |
.beta.-Alanyl thio esters Gil Clifton and Charles G. Skinner pp 575 - 577; DOI: 10.1021/jm00297a068 |
Metal complexes of 1-substituted 3-hydroxyureas Robert E. Harmon, James C. Dabrowiak, Donald John Brown, Surendra Kumar Gupta, Michael Herbert, and Dakshinamurthy Chitharanjan pp 577 - 579; DOI: 10.1021/jm00297a069 |
Potential antineoplastics. III. Series of 1-thiocarbamoyl-3-methyl-4-arylazo-5-methyl(or phenyl)pyrazoles Hari G. Garg and Ram Ashrey Sharma pp 579 - 581; DOI: 10.1021/jm00297a070 |
Synthesis of mono-, di-, and trimethoxy derivatives of N,N-bis(2-chloroethyl)aniline and related compounds as antitumor agents A. H. Sommers, Ursula Biermacher, Sandra B. Brehm, and James H. Short pp 581 - 583; DOI: 10.1021/jm00297a071 |
Benzylidene hydrazides as potential anticancer agents David W. Boykin and Rajendra S. Varma pp 583 - 584; DOI: 10.1021/jm00297a072 |
Substituted [p-(p-ethoxyphenyl)anilino]acetamides Giovanni Brancaccio, G. Lettieri, Angelo Larizza, Rene Viterbo, and G. C. Perri pp 584 - 584; DOI: 10.1021/jm00297a073 |
Substituted chroman-6-ylureas and thioureas G. Lettieri, Giovanni Brancaccio, Angelo Larizza, and Rene Viterbo pp 584 - 585; DOI: 10.1021/jm00297a074 |
The Biochemistry of Viruses Alfred Burger pp 586 - 586; DOI: 10.1021/jm00297a900 |
Proceedings of the Institute on Drug Literature Evaluation Maxwell Gordon pp 586 - 586; DOI: 10.1021/jm00297a901 |
The Chemistry and Biochemistry of Steroids Manfred E. Wolff pp 586 - 586; DOI: 10.1021/jm00297a902 |
Synthetic schistosomicides. XVII. N-(Benzylidene and cinnamylidene)-N'-[2-(diethylamino)ethyl]-1,4-naphthalenediamines and related Schiff bases Edward F. Elslager, Josephine Battaglia, Annette A. Phillips, and Leslie M. Werbel pp 587 - 592; DOI: 10.1021/jm00298a001 |
Synthetic schistosomicides. XVIII. N-(4-[[2-(Diethylamino)ethyl]amino]-1-naphthyl)amides, N-[5,6,7,8-tetrahydro-4-[(3-piperidinopropyl)amino]-1-naphthyl]amides, and related amide and urea derivatives Leslie M. Werbel, Josephine Battaglia, Edward F. Elslager, and Carl Youngstrom pp 592 - 598; DOI: 10.1021/jm00298a002 |
Synthesis and schistosomicidal activity of 6-chloro-5-[[2-(diethylamino)ethyl]amino]-8-quinolinemethanol Denis M. Bailey, Sydney Archer, David Wood, David Rosi, and Allen Yarinsky pp 598 - 601; DOI: 10.1021/jm00298a003 |
Coenzyme Q. CXXII. Identification and ubiquinone-8 biosynthesized by Plasmodium knowlesi, P. cynomolgi, and P. berghei Frederick S. Skelton, P. J. Rietz, and Karl Folkers pp 602 - 606; DOI: 10.1021/jm00298a004 |
Acyloxymethyl esters of ampicillin Wolf Von Daehne, E. Frederiksen, E. Gundersen, F. Lund, P. Moerch, Hans J. Petersen, Knud Roholt, L. Tybring, and Wagn O. Godtfredsen pp 607 - 612; DOI: 10.1021/jm00298a005 |
Isoquinolines. 1. 3-Amino- and 3-fluoroisoquinoline derivatives as potential antimalarials John L. Neumeyer and Klaus K. Weinhardt pp 613 - 616; DOI: 10.1021/jm00298a006 |
Lincomycin. XI. Synthesis and structure of clindamycin, a potent antibacterial agent Robert D. Birkenmeyer and Fred Kagan pp 616 - 619; DOI: 10.1021/jm00298a007 |
Antiviral phenoxathiins and their analogs. Study of the structure-activity relations for antiviral activity and the replacement ability in poliovirus type III dependent variants Charles J. Paget, Earleen M. Dennis, Janet Nelson, and Donald C. DeLong pp 620 - 623; DOI: 10.1021/jm00298a008 |
Structure-activity correlations for the central nervous system depressant 2-imidazolidinones Eric J. Lien, Mehdi Hussain, and Michael P. Golden pp 623 - 626; DOI: 10.1021/jm00298a009 |
Stereochemical studies on medicinal agents. VIII. Absolute stereochemistries of isomethadol isomers Philip S Portoghese and David Allen Williams pp 626 - 630; DOI: 10.1021/jm00298a010 |
Homologs of benzomorphan derivatives. 1 Mikio Takeda and Hiroshi Kugita pp 630 - 634; DOI: 10.1021/jm00298a011 |
Preparation of substituted naphthylcyclohexane derivatives and related compounds Humberto Carpio, Wendell H. Rooks, and Pierre Crabbe pp 634 - 637; DOI: 10.1021/jm00298a012 |
Nitrofuryl heterocyclics. 1 M. D. Closier and Peter J. Islip pp 638 - 640; DOI: 10.1021/jm00298a013 |
Synthesis and pharmacology of N-cyano-(.beta.-arylethyl)amines Edward E. Smissman, Alexandros C. Makriyannis, and Edward J. Walaszek pp 640 - 644; DOI: 10.1021/jm00298a014 |
Piperidine derivatives. 1 Michio Nakanishi, Chiaki Tashiro, Tomohiko Munakata, Kazuhiko Araki, Tatsumi Tsumagari, and Hiroshi Imamura pp 644 - 648; DOI: 10.1021/jm00298a015 |
Synthesis and pharmacological activity of new basic carbamates Georges Tsatsas, Aspasia Papadakis-Valirakis, Wilbur M. Benson, and Samuel A. Ferguson pp 648 - 651; DOI: 10.1021/jm00298a016 |
Acetylene compounds of potential pharmacological value. XIV. N-(tert-aminoalkynyl)-substituted succinimides and maleimides. Class of central anticholinergic agents Bo Karlen, Bjorn Lindeke, Sune Lindgren, Karl G. Svensson, Richard Dahlbom, Donald J. Jenden, and John E. Giering pp 651 - 657; DOI: 10.1021/jm00298a017 |
Modified cardenolides. V. Replacement of the C-17 lactone substituent by alkylating groups Manfred E. Wolff, Hong-Hsi Chang, and Winston Ho pp 657 - 663; DOI: 10.1021/jm00298a018 |
Basic ethers of 1-(p-hydroxyphenyl)-2-phenyl-1,2,3,4-tetrahydroquinoline and 1-(p-hydroxyphenyl)-2-phenylindole. Antifertility agents Malcolm Rice Bell, Andrew W. Zalay, Rudolf Oesterlin, Philip Schane, and Gordon O. Potts pp 664 - 668; DOI: 10.1021/jm00298a019 |
Synthesis and antiarrhythmic activity of naphthylalkylamines Gianfranco Pala, Arturo Donetti, Carla Turba, and Silvano Casadio pp 668 - 671; DOI: 10.1021/jm00298a020 |
4-Alkyl-5-aryl-4H-1,2,4-triazole-3-thiols as hypoglycemic agents M. Y. Mhasalkar, Madhusudan H. Shah, S. T. Nikam, Kodaganallur G. Anantanarayanan, and Chimanlal V. Deliwala pp 672 - 674; DOI: 10.1021/jm00298a021 |
Saligenin analogs of sympathomimetic catechol amines David T. Collin, David Hartley, David Jack, Lawrence H. C. Lunts, J. C. Press, Alexander C. Ritchie, and Paul Toon pp 674 - 680; DOI: 10.1021/jm00298a022 |
Inhibition of serotonin[3H] uptake by the mouse spleen. Structure-activity study Robert A. Lahti, Patricia A. Platz, and Barbara J. McAllister pp 681 - 683; DOI: 10.1021/jm00298a023 |
Derivatives of 3,4-dihydro-1(2H)-naphthalenone as .beta.-adrenergic blocking agents. 1. Bunolol and related analogs Charles F. Schwender, Sheldon Farber, Carol Blaum, and John Shavel pp 684 - 688; DOI: 10.1021/jm00298a024 |
Ionization of histamine, N-acetylhistamine, and their iodinated derivatives T. B. Paiva, Mineko Tominaga, and Antonio C. M. Paiva pp 689 - 692; DOI: 10.1021/jm00298a025 |
Potential coenzyme inhibitors. IV. 3-Acetyl substituted pyridine and dihydropyridine derivatives Andrew C. Lovesey pp 693 - 696; DOI: 10.1021/jm00298a026 |
Neuraminidase inhibition and viral chemotherapy Theodore H. Haskell, Floyd E. Peterson, Donald Watson, Nike R. Plessas, and Townley Culbertson pp 697 - 704; DOI: 10.1021/jm00298a027 |
Synthesis and pharmacological evaluation of some pyridylmethyl substituted ethylenediamines Seiji Miyano, Akiko Abe, Yoshitoshi Kase, Tomokazu Yuizono, Kuniomi Tachibana, Takeshi Miyata, and Go Kito pp 704 - 708; DOI: 10.1021/jm00298a028 |
Synthesis of 5-mercaptouridine Gabor L. Szekeres and Thomas J. Bardos pp 708 - 712; DOI: 10.1021/jm00298a029 |
Novel polycyclic heterocycles. Derivatives of 5,11-dihydrodibenz[b,e][1,4]oxazepine and 5,11-dihydrodibenzo[b,e][1,4]thiazepine Harry L. Yale, Bernard Beer, Jelka Pluscec, and Erwin R. Spitzmiller pp 713 - 722; DOI: 10.1021/jm00298a030 |
Synthesis and hypocholesterolemic activity of alkylidenedithio bisphenols Martin B. Neuworth, Rohert J. Laufer, James W. Barnhart, J. A. Sefranka, and D. D. McIntosh pp 722 - 725; DOI: 10.1021/jm00298a031 |
Synthesis and antiinflammatory activity of some aryltetrazolylalkanoic acids Robert T. Buckler, Shin Hayao, O. J. Lorenzetti, Lawrence F. Sancilio, Harold E. Hartzler, and Wallace G. Strycker pp 725 - 729; DOI: 10.1021/jm00298a032 |
Synthesis and screening for antideperessant activity of some aminoindanooxazolines, aminoindanooxazines, and aminoacenaphthoxazolines Donald L. Trepanier, H. Eldridge Faith, and John N. Eble pp 729 - 733; DOI: 10.1021/jm00298a033 |
Chemotherapeutic nitroheterocycles. 1. Substituted 2-(5-nitro-2-furyl)pyrimidines Rudolf Albrecht, Klaus Gutsche, Hans J. Kessler, and Eberhard Schroeder pp 733 - 735; DOI: 10.1021/jm00298a034 |
Chemotherapeutic nitroheterocycles. 2. 2-(5-Nitro-2-furyl)pyrimidines with basic substituents Rudolf Albrecht, Klaus Gutsche, Hans J. Kessler, and Eberhard Schroeder pp 736 - 737; DOI: 10.1021/jm00298a035 |
Reassignment of the absolute configuration of 3-acetoxyquinuclidine methiodide and the absolute configuration of receptor-bound acetylcholine Bernard Belleau and Peter Pauling pp 737 - 738; DOI: 10.1021/jm00298a036 |
Synthesis of compounds related to muscimol (pantherine, agarin) Bernard Loev, James William Wilson, and Marjorie M. Goodman pp 738 - 741; DOI: 10.1021/jm00298a037 |
Benzimidazole-5(6)-alanine and related compounds. I. Synthesis of amino acids as inhibitors of norepinephrine biosynthesis John D. Milkowski, Francis M. Miller, Eugene M. Johnson, and Nicolas Zenker pp 741 - 742; DOI: 10.1021/jm00298a038 |
Synthesis and structure-activity relations of 1-alkoxyalkyl- and 1-aryloxyalkyl-1,4-benzodiazepin-2-ones Samuel Lamdan, C. H. Gaozza, S. Sicardi, and J. A. Izquierdo pp 742 - 744; DOI: 10.1021/jm00298a039 |
Angiotensin II analogs. IV. Synthesis and biological evaluation of simplified angiotensins Eugene C. Jorgensen, Graham C. Windridge, and Thomas Choy Lee pp 744 - 745; DOI: 10.1021/jm00298a040 |
Thyroxine analogs. XIX. 3,5-Dimethyl-3'-isopropyl-DL-thyronine Eugene C. Jorgensen and Jeremy Wright pp 745 - 747; DOI: 10.1021/jm00298a041 |
Central nervous system activity of ethyl 1-naphthylalkylcarbamates Arturo Donetti and Ernesta Marazzi-Uberti pp 747 - 748; DOI: 10.1021/jm00298a042 |
Synthesis and endocrine activity of some 3-aza-A-homopregnenes Arvin P. Shroff pp 748 - 750; DOI: 10.1021/jm00298a043 |
Preparation of 6-acetamino-16-methylene-17.alpha.-hydroxy-4,6-pregnadiene-3,20-dione 17-acetate G. Teutsch, Elliot L. Shapiro, and Hershel L. Herzog pp 750 - 751; DOI: 10.1021/jm00298a044 |
Ring-D-bridged steroid analogs. VIII. Testosterone analogs Alan J. Solo, J. N. Kapoor, and Peter Hebborn pp 751 - 754; DOI: 10.1021/jm00298a045 |
Analogs of steroid hormones. IV. 16-Keto steroid derivatives Richard E. Juday and Bonnie Bukwa pp 754 - 755; DOI: 10.1021/jm00298a046 |
Potential specific inhibitors of the lactose transport system of Escherichia coli Emrys Wyn Thomas pp 755 - 756; DOI: 10.1021/jm00298a047 |
1-Substituted 3-[(5-nitrofurfurylidene)amino]-2-imidazolidinones Harry R. Snyder, Frank F. Ebetino, A. J. Siedler, and Jon Andersen pp 756 - 759; DOI: 10.1021/jm00298a048 |
Antimalarial sulfilimines and sulfoximines related to diaminodiphenyl sulfoxide and sulfone Kenneth K. Andersen, Jnanabrata Bhattacharyya, and Sunil K. Mukhopadhyay pp 759 - 760; DOI: 10.1021/jm00298a049 |
Synthesis and antimalarial activity of 4-aminobenzo[g-1,5]naphthyridines Ned D. Heindel and Stephen A. Fine pp 760 - 762; DOI: 10.1021/jm00298a050 |
Synthesis and antineoplastic evaluation of some 9-substituted acridines James Thomas Stewart and David M. Shepherd pp 762 - 762; DOI: 10.1021/jm00298a051 |
Potential antineoplastics. IV. 2-Amino-4-methyl-6-phenyl-5-arylazopyrimidines Hari G. Garg and Ram Ashrey Sharma pp 763 - 765; DOI: 10.1021/jm00298a052 |
Synthesis of 5-iodo-3-indolylphosphodiesters of 5-fluorodeoxyuridine as possible chromogenic cancer chemotherapeutic agents Kwan-Chung Tsou, Shohei Aoyagi, and Elizabeth Eshelman Miller pp 765 - 768; DOI: 10.1021/jm00298a053 |
Structure-antitumor activity correlation of some Schiff bases Ernest M. Hodnett and William J. Dunn pp 768 - 770; DOI: 10.1021/jm00298a054 |
Antineoplastic research. I. Pyrazole and pyrimidine derivatives of dehydrocycloheximide analogs David M. Piatak, C. C. Yen, and R. V. Kennedy pp 770 - 771; DOI: 10.1021/jm00298a055 |
Halogenated 1-(4-aminobenzylidene)indenes Carl T. Bahner, David H. Brotherton, Jane Cline, Harold Kinder, and Lydia M. Rives pp 771 - 773; DOI: 10.1021/jm00298a056 |
Synthesis and alkylation of tetrahydrocyclopentapyrazolols Richard P. Williams, Victor J. Bauer, and Sidney R. Safir pp 773 - 775; DOI: 10.1021/jm00298a057 |
Puromycin analogs. Aminoacyl derivatives of 9-(3'-amino-3'-deoxy-.beta.-D-arabino-furanosyl)adenine Linda V. Fisher, William W. Lee, and Leon Goodman pp 775 - 777; DOI: 10.1021/jm00298a058 |
Alkylation of 5-substituted tetrazoles Leland Huff and Ronald A. Henry pp 777 - 779; DOI: 10.1021/jm00298a059 |
Aminoadamantane derivatives as potential insect chemosterilants James E. Oliver and Jerry B. Stokes pp 779 - 780; DOI: 10.1021/jm00298a060 |
Potential antidiabetics. V. 3,5-Dimethyl-4-arylazo-N1-carbamoyl-, 3-methyl-4-arylazo-5-phenyl-N1-carbamoyl-, and 3,5-dimethyl-4-arylazo-N1-hippurylpyrazoles Wahid U. Malik, Hari G. Garg, Prem P. Singh, and Veena Arora pp 780 - 782; DOI: 10.1021/jm00298a061 |
Insect chemosterilants. IX. N-(Hydroxymethyl)-N,N',N',N'',N''-pentamethylphosphoric triamide Paul H. Terry and Alexej B. Borkovec pp 782 - 783; DOI: 10.1021/jm00298a062 |
New thio derivatives of carcinogenic arylamines. IV. 4-Acetamido-3-methylthiodiphenyl T. Lloyd Fletcher, Carol A. Cole, Hsi-Lung Pan, and Moses J. Namkung pp 784 - 784; DOI: 10.1021/jm00298a063 |
New benzimidazoles William R. Sullivan pp 784 - 786; DOI: 10.1021/jm00298a064 |
Antitumor activities of some Schiff bases Ernest M. Hodnett and Paul D. Mooney pp 786 - 786; DOI: 10.1021/jm00298a065 |
The Chemistry of the Isoquinoline Alkaloids Tetsuji Kametaxi pp 787 - 787; DOI: 10.1021/jm00298a900 |
Advances in Biochemical Psychopharmacology Alfred Burger pp 787 - 787; DOI: 10.1021/jm00298a901 |
Hormonal Contraception Manfred E. Wolff pp 787 - 787; DOI: 10.1021/jm00298a902 |
Strcutural Units of Medical and Biological Terms. A Convenient Guide, in English, to the Roots, Stems, Prefixes, Suffixes, and Other Combining Forms which are the Building Blocks of Medical and Related Scientific Words Alfred Burger pp 787 - 787; DOI: 10.1021/jm00298a903 |
The National Formulary Alfred Burger pp 788 - 788; DOI: 10.1021/jm00298a904 |
Synthetic Methods of Organic Chemistry Richard J. Sundberg pp 788 - 788; DOI: 10.1021/jm00298a905 |
Thiamine Diphosphate and Its Catalytic Functions Alfred Burger pp 788 - 788; DOI: 10.1021/jm00298a906 |
Fondamenti di Chimica Farmaceutica R. Deghenghi pp 788 - 788; DOI: 10.1021/jm00298a907 |
Synthesis of .gamma.-dimethylaminomethyl-.alpha.-phenylcycloalkyl propionates as potential analgetics Mathias P. Mertes, Arthur A. Ramsey, Patrick E. Hanna, and Duane D. Miller pp 789 - 794; DOI: 10.1021/jm00299a001 |
Analgetics based on the pyrrolidine ring. V John F. Cavalla, Ian M. Lockhart, Nigel E. Webb, Claude V. Winder, Myrna Welford, and Agnes Wong pp 794 - 800; DOI: 10.1021/jm00299a002 |
Structure-activity correlations of morphinelike analgetics based on efficiencies following intravenous and intraventricular application Eberhard Kutter, Albert Herz, Hans J. Teschemacher, and Rainer Hess pp 801 - 805; DOI: 10.1021/jm00299a003 |
Optical isomers of miscellaneous strong analgetics Everette L. May and Mikio Takeda pp 805 - 807; DOI: 10.1021/jm00299a004 |
Tricyclic norephedrine analogs. Isomeric 9-hydroxy-10-amino-1,2,3,4,4a,9,10,10a-(trans-4a,10a)-octahydrophenanthrenes Wendel Lane Nelson and Duane D. Miller pp 807 - 814; DOI: 10.1021/jm00299a005 |
Synthesis and hypotensive activity of N-substituted 1-trimethoxybenzyl-3-butenylamines and related compounds F. J. McCarty, L. J. Lendvay, A. J. Vazakas, W. W. Bennetts, F. P. Palopoli, R. Orzechowski, and S. Goldstein pp 814 - 819; DOI: 10.1021/jm00299a006 |
Synthesis and anorectic activity of some 1-benzylcyclopropylamines Carl Kaiser, Charles A. Leonard, George C. Heil, Bruce M. Lester, David H. Tedeschi, and Charles L. Zirkle pp 820 - 826; DOI: 10.1021/jm00299a007 |
Pyrrolo[3,2,1-jk][1,4]benzodiazepines and pyrrolo[1,2,3-ef][1,5]benzodiazepines which have central nervous system activity Jackson B. Hester, Allan D. Rudzik, and William Veldkamp pp 827 - 835; DOI: 10.1021/jm00299a008 |
4-Substituted piperidines. V. Local anesthetic 4-aminoalkoxy-4-arylpiperidines Bert Hermans, Hugo Verhoeven, and Paul Janssen pp 835 - 838; DOI: 10.1021/jm00299a009 |
Polypeptides. XLVI. Synthesis of a stably labeled, biologically active adrenocorticotropin fragment Luis Moroder and Klaus Hofmann pp 839 - 843; DOI: 10.1021/jm00299a010 |
Synthesis of pyroglutamylhistidylprolineamide by classical and solid phase methods George Flouret pp 843 - 845; DOI: 10.1021/jm00299a011 |
N-Aminoalkylpolyglycine. Synthesis, antibacterial activity, and electrochemical behavior as a titrant of living cells Eleonora Santucci, Marcello Marchetti, Franco Alhaique, Claudio Botre, and Fulvio M. Riccieri pp 846 - 848; DOI: 10.1021/jm00299a012 |
Alkylation of 2-methyl-5-nitroimidazole. Some potent antiprotozoal agents Max Warren Miller, Harold L. Howes, Robert V. Kasubick, and Arthur R. English pp 849 - 852; DOI: 10.1021/jm00299a013 |
Synthesis of potential antimalarial agents. V. Pyrido[2,3-b]pyrazines Carroll Temple, Jerry D. Rose, Robert Daryl Elliott, and John A. Montgomery pp 853 - 857; DOI: 10.1021/jm00299a014 |
In vivo hydrolysis of isomeric bis(1,1,1-trichloro-2-propyl)1,2-cyclobutanedicarboxylates Jorge P. Li, John H. Biel, Donald R. Van Harken, Lorraine T. Harmanos, Clarence W. Dixon, and Harold D. Taylor pp 858 - 859; DOI: 10.1021/jm00299a015 |
Antimalarials. II. 8-Quinolinemethanols J. Samuel Gillespie, Satya P. Acharya, Richard E. Davis, and B. K. Barman pp 860 - 864; DOI: 10.1021/jm00299a016 |
New synthesis of antimalarials related to 2-bromo-4,5-dimethoxy-N,N-bis(diethylaminoethyl)aniline. Terminal nitrogen modifications Eugene L. Strogryn pp 864 - 866; DOI: 10.1021/jm00299a017 |
Structural modification of febrifugine. Some methylenedioxy analogs Ping-Lu Chien and Chia-Chung Cheng pp 867 - 870; DOI: 10.1021/jm00299a018 |
Structure and anticoccidial activity among some 4-hydroxyquinolinecarboxylates Renat H. Mizzoni and et al. pp 870 - 878; DOI: 10.1021/jm00299a019 |
Anticoccidial activity in 1-[2-(cycloalkyl)- and 2-(cycloalkylmethyl-4-amino-5-pyrimidyl)methyl]pyridinium salts Renat H. Mizzoni and et al. pp 878 - 882; DOI: 10.1021/jm00299a020 |
Quinazolines. VI. Synthesis of 2,4-diaminoquinazolines from anthranilonitriles Andre Rosowsky, James L. Marini, Marilyn E. Nadel, and Edward J. Modest pp 882 - 886; DOI: 10.1021/jm00299a021 |
Synthesis and activity of some 3-aryl- and 3-aralkyl-1,2,3,4-tetrahydro-4-oxo-6-quinazolinesulfonamides Bola V. Shetty, Liborio A. Campanella, Telfer L. Thomas, M. Fedorchuk, T. A. Davidson, L. Michelson, H. Volz, S. E. Zimmerman, E. J. Belair, and A. P. Truant pp 886 - 895; DOI: 10.1021/jm00299a022 |
Aminoalkenylbenzenesulfonamides with hypotensive and histamine-releasing properties Marion T. Dorsett, J. Martin Grisar, Kenneth R. Hickey, Rudolph L. Pohl, William J. Hudak, and Richard E. Lewis pp 895 - 900; DOI: 10.1021/jm00299a023 |
Comparative effects of piperonyl butoxide and N-(4-pentynyl)phthalimide on mammalian microsomal enzyme functions Herbert Jaffe and John L. Neumeyer pp 901 - 903; DOI: 10.1021/jm00299a024 |
In vivo hydroxylation of the alkaloid acronine, an experimental antitumor agent Hugh Richard Sullivan, Ruth E. Billings, John L. Occolowitz, Harold E. Boaz, Frederick J. Marshall, and Robert E. McMahon pp 904 - 909; DOI: 10.1021/jm00299a025 |
Choline acetyltransferase inhibitors. Physicochemical properties in relation to inhibitory activity of styrylpyridine analogs Richard Charles Allen, Gerald L. Carlson, and C. J. Cavallito pp 909 - 912; DOI: 10.1021/jm00299a026 |
Structure-activity relations in thymidine phosphorylase inhibitors. A correlation using substituent constants and regression analysis Eugene Coats, W. R. Glave, and Corwin Hansch pp 913 - 919; DOI: 10.1021/jm00299a027 |
Mixed bifunctionality. III. Antitumor activity of sesame oil solutions of simple alkylating derivatives of polynuclear hydrocarbons Richard M. Peck and Anna P. O'Connell pp 919 - 922; DOI: 10.1021/jm00299a028 |
Electron-donating properties of phenothiazine and related compounds John E. Bloor, Bruce R. Gilson, R. J. Haas, and Charles L. Zirkle pp 922 - 925; DOI: 10.1021/jm00299a029 |
Bridged bicyclic and polycyclic amino acids. Potent new inhibitors of the fibrinolytic process Larry J. Loeffler, Susan F. Britcher, and Werner Baumgarten pp 926 - 935; DOI: 10.1021/jm00299a030 |
Potential anticancer agents. III. Schiff bases from benzaldehyde nitrogen mustards and aminophenylthiazoles J. D. Modi, S. S. Sabnis, and C. V. Deliwala pp 935 - 941; DOI: 10.1021/jm00299a031 |
Synthesis of dideoxyzearalanone and hydroxyl derivatives David B. R. Johnston, Carol A. Sawicki, Thomas B. Windholz, and A. A. Patchett pp 941 - 944; DOI: 10.1021/jm00299a032 |
Relation between lipophilic character and hemolytic activity of testosterone and testosterone esters Gian L. Biagi, Maria C. Guerra, and Anna M. Barbaro pp 944 - 948; DOI: 10.1021/jm00299a033 |
Steroidal heterocycles. XIII. 4.alpha.,5-Epoxy-5.alpha.-androst-2-eno[2,3-d]isoxazoles and related compounds H. C. Neumann, G. O. Potts, W. T. Ryan, and F. W. Stonner pp 948 - 951; DOI: 10.1021/jm00299a034 |
Anabolic 19-nortestosterone bicyclo[2.2.2]octane- and -octenecarboxylates Richard M. Scribner, R. I. Dorfman, and W. H. Rooks pp 952 - 956; DOI: 10.1021/jm00299a035 |
Role of the benzyl moiety in biochemical and pharmacological processes Corwin Hansch and Richard Kerley pp 957 - 964; DOI: 10.1021/jm00299a036 |
Use of .sigma.+ in structure-activity correlations Corwin Hansch pp 964 - 966; DOI: 10.1021/jm00299a037 |
Metal chelate steroid analog. [7-Amino-3-(1,5-dimethylhexyl)dodecahydro-3a,6-dimethyl-1H-benz[e]indene-6-methylamine]bis(ethylenediamine)cobalt(3 +) trichloride Lorraine G. Donaruma and Patricia U. Flath pp 966 - 967; DOI: 10.1021/jm00299a038 |
Synthesis and myotrophic-androgenic activity of 17.beta.-hydroxy-5.alpha.-androst-8(14)-en-3-one derivatives Manfred Ernst Wolff and Hong-Hsi Chang pp 967 - 968; DOI: 10.1021/jm00299a039 |
Imidazole derivatives. Histidine decarboxylase inhibitors Leo R. Swett and Tobias O. Yellin pp 968 - 970; DOI: 10.1021/jm00299a040 |
New .beta.-adrenergic blocking agents. Cyclopropylphenyl derivatives Jacques R. Boissier, Roger Ratouis, Claude Dumont, Pierre H. Derible, and Jean P. Lavaux pp 971 - 973; DOI: 10.1021/jm00299a041 |
2,3,6-Trimethoxynitrostyrene and its .beta.-phenethylamine Betty Matsuhiro and Arthur Furst pp 973 - 973; DOI: 10.1021/jm00299a042 |
Synthesis of B/C trans-fused morphine structures. V. Pharmacological summary of trans-morphine derivatives and an improved synthesis of trans-codeine Hiroshi Kugita, Mikio Takeda, and Hirosumi Inoue pp 973 - 975; DOI: 10.1021/jm00299a043 |
Analeptics. 1-Formimidoylindolines Yao-Hua Wu, Walter G. Lobeck, and John W. Kissel pp 975 - 977; DOI: 10.1021/jm00299a044 |
Synthesis of some local anesthetics Pramod K. Srivastava and P. N. Srivastava pp 977 - 979; DOI: 10.1021/jm00299a045 |
Synthesis of some substituted 10-amino-10,11-dihydro-5H-dibenz[b,f]azepines Bijan Prasun Das, Ronald W. Woodard, Larry K. Whisenant, William F. Winecoff, and David W. Boykin pp 979 - 981; DOI: 10.1021/jm00299a046 |
New class of 1,3-benzoxazinones as potential central nervous system agents Ned D. Heindel and Lee A. Schaeffer pp 981 - 983; DOI: 10.1021/jm00299a047 |
Substituted oxindoles. III. Synthesis and pharmacology of some substituted oxindoles John Walker, Roy W. Daisley, and Arnold H. Beckett pp 983 - 985; DOI: 10.1021/jm00299a048 |
Demethylation studies. VII. Unique effect of the N-cyclopropyl group in a new series of inhibitors of oxidative microsomal demethylation Robert E. McMahon, Hilman W. Culp, and Jack Mills pp 986 - 987; DOI: 10.1021/jm00299a049 |
Pyrazine diuretics. VIII. N-Amidino-3-aminopyrazinecarboxamide 4-oxides James Holden Jones and Edward J. Cragoe pp 987 - 989; DOI: 10.1021/jm00299a050 |
Modification of recovered dominant lethal mutations induced by heteroaromatic aziridines in stored housefly sperm J. George Pomonis, David T. North, and Richard G. Zaylskie pp 989 - 991; DOI: 10.1021/jm00299a051 |
Potential antineoplastics. V. Synthesis of ethyl 2,3-dioxobutyrate 2-arylhydrazono-3-thiosemicarbazones Hari G. Garg and Ram Ashrey Sharma pp 991 - 992; DOI: 10.1021/jm00299a052 |
Quaternary indolylpyridinium salts. Oral hypoglycemic agents William J. Fanshawe, Victor J. Bauer, Sidney R. Safir, D. A. Blickens, and S. J. Riggi pp 993 - 995; DOI: 10.1021/jm00299a053 |
Folic acid analogs. II. p-{[(2,6-Diamino-8-purinyl)methyl]amino}-benzoyl-L-glutamic acid and related compounds Louis T. Weinstock, Bernard F. Grabowski, and Chia-Chung Cheng pp 995 - 997; DOI: 10.1021/jm00299a054 |
Sodium tyropanoate, a new oral cholecystographic agent J. O. Hoppe, J. H. Ackerman, A. A. Larsen, and J. Moss pp 997 - 999; DOI: 10.1021/jm00299a055 |
Isoquinolines. 2. 3-(Dialkylaminoalkylamino)isoquinolines as potential antimalarial drugs John L. Neumeyer and Klaus K. Weinhardt pp 999 - 1002; DOI: 10.1021/jm00299a056 |
Antimalarial agents. VI. 5-Quinolinemethanols Ivan C. Popoff and Chandrakant B. Thanawalla pp 1002 - 1004; DOI: 10.1021/jm00299a057 |
Potential antimalarials. V. 2-p-Chlorophenyl-7-quinolinemethanols Lee C. Washburn, T. G. Barbee, and D. E. Pearson pp 1004 - 1005; DOI: 10.1021/jm00299a058 |
Quinoxaline studies. XVII. Potential antimalarials. Some (RS)-.alpha.-(dialkylaminomethyl)-6-chloro-2-quinoxalinemethanols Henry R. Moreno and Harry P. Schultz pp 1005 - 1008; DOI: 10.1021/jm00299a059 |
Synthesis and antimicrobial activity of 5,7-dichloroquinoline-8-thiol and its derivatives Alan O. Fitton and Frank Ridgway pp 1008 - 1009; DOI: 10.1021/jm00299a060 |
Structural modification studies of 3-piperonylsydnone. 2. Synthesis of piperonyl-substituted hydantoin, thiohydantoin, thiazolidinedione, rhodanine, imidazolinone, and related compounds William H. Burton, William L. Budde, and Chia-Chung Cheng pp 1009 - 1012; DOI: 10.1021/jm00299a061 |
In vivo antiviral effects of benzothiazole derivatives against various influenza A2 strains Stig Akerfeldt pp 1012 - 1013; DOI: 10.1021/jm00299a062 |
Cycloserine derivatives Charles H. Stammer, C. Chandrasekharan Kartha, Nishith C. Chaturvedi, and James D. McKinney pp 1013 - 1015; DOI: 10.1021/jm00299a063 |
Nitroheterocyclic antimicrobial agents. II. 5-Nitro-1,3,4-thiadiazole-2-carboxaldehyde derivatives Goro Asato, Gerald Berkelhammer, and Edward L. Moon pp 1015 - 1017; DOI: 10.1021/jm00299a064 |
Indole derivatives Frank D. Popp pp 1017 - 1018; DOI: 10.1021/jm00299a065 |
Chemistry of azole derivatives. XII. Possible anticonvulsant thiazolo[3,2-a]benzimidazoles Jag Megh Singh pp 1018 - 1018; DOI: 10.1021/jm00299a066 |
Reinvestigation of the reaction of monosodium urea with various substituted pyrazinecarboxylate esters J. William Hanifin, Rosemary Capuzzi, and Elliott Cohen pp 1018 - 1019; DOI: 10.1021/jm00299a067 |
N-Aryl-N-aroylamino acid derivatives A. Larizza, G. Lettieri, and R. Viterbo pp 1019 - 1020; DOI: 10.1021/jm00299a068 |
Ferrocene studies. V. Potential medicinal agents Frank D. Popp and E. Bradley Moynahan pp 1020 - 1021; DOI: 10.1021/jm00299a069 |
Bis(.alpha.-lactams) derived from adamantane Erach R. Talaty and Aubry E. Dupuy pp 1021 - 1022; DOI: 10.1021/jm00299a070 |
Derivatives of 2,5-dimethoxy-4-methylamphetamine (DOM) Beng-Thong Ho, L. Wayne Tansey, and William M. McIsaac pp 1022 - 1022; DOI: 10.1021/jm00299a071 |
1-Substituted 2,5-dimethylpyrroles Laird F. Miller and Ronald E. Bambury pp 1022 - 1023; DOI: 10.1021/jm00299a072 |
Newer cardiac glycosides and aglycones Ko Kuei Chen pp 1029 - 1034; DOI: 10.1021/jm00300a001 |
Supplementary glycosides of digitalis Ko Kuei Chen pp 1035 - 1037; DOI: 10.1021/jm00300a002 |
Small ring analogs of acetylcholine. Synthesis and absolute configurations of cyclopropane derivatives Joseph G. Cannon and Paul Douglas Armstrong pp 1037 - 1039; DOI: 10.1021/jm00300a003 |
Aromatic amino acid hydroxylase inhibitors. I. Halogenated phenylalanines Raymond E. Counsell, P. Desai, Terry Douglas Smith, Peter S. Chan, P. A. Weinhold, V. B. Rethy, and D. Burke pp 1040 - 1042; DOI: 10.1021/jm00300a004 |
Inhibition of adrenal phenethanolamine N-methyltransferase by substituted benzimidazoles Lewis R. Mandel, Curt Culwell Porter, F. A. Kuehl, N. P. Jensen, S. M. Schmitt, T. B. Windholz, T. R. Beattie, J. A. Carty, B. G. Christensen, and Tsung-Ying Shen pp 1043 - 1047; DOI: 10.1021/jm00300a005 |
Imidazole derivatives. IV. Synthesis and pharmacologic activity of oxygenated derivatives of imidazo[1,2-a]pyridine Luigi Almirante, Alfonso Mugnaini, Nicola De Toma, Afro Gamba, Walter Murmann, and John Hidalgo pp 1048 - 1051; DOI: 10.1021/jm00300a006 |
Aralkylaminoguanidines and related compounds John B. Bream, Claude W. Picard, Trevor G. White, and Hans Lauener pp 1051 - 1057; DOI: 10.1021/jm00300a007 |
Synthesis and norepinephrine depleting activity of some metaraminol ethers Walfred S. Saari, Andrew W. Raab, William H. Staas, M. L. Torchiana, Curt Culwell Porter, and Clement Addison Stone pp 1057 - 1061; DOI: 10.1021/jm00300a008 |
Agonists-antagonists derived from desomorphine and metopon Lewis J. Sargent and Everette L. May pp 1061 - 1063; DOI: 10.1021/jm00300a009 |
Syntheses of heterocyclic compounds. CCCLXXX. Azamorphinan and related compounds. III. Syntheses of 3-hydroxy-N-substituted-9-azamorphinans Tetsuji Kametani, Kazuo Kigasawa, Mineharu Hiiragi, Nagatoshi Wagatsuma, Kikuo Wakisaka, Fumio Satoh, and Setsu Saito pp 1064 - 1067; DOI: 10.1021/jm00300a010 |
Potential antiinflammatory agents. Aralkoxyhydrouracils and aralkoxyhydantoins Leon Simet, D. B. Reisner, Bernard J. Ludwig, F. Duersch, and Frank Milan Berger pp 1067 - 1071; DOI: 10.1021/jm00300a011 |
Aminobenzoic acid diuretics. 1. 4-Halogeno-5-sulfamylmetanilic acid derivatives Peter W. Feit, Herta Bruun, and Christian K. Nielsen pp 1071 - 1075; DOI: 10.1021/jm00300a012 |
Spasmolytics. II. 3-Tropanyl 2,3-diarylacrylates Henry C. Caldwell, Joseph A. Finkelstein, Philip P. Goldman, Andrew J. Sivak, Jack Schlosser, Carol Pelikan, and William G. Groves pp 1076 - 1079; DOI: 10.1021/jm00300a013 |
Spasmolytics. III. 3-Tropanyl 2,3-diarylacrylates. Case history of .pi.-.sigma. structure-function correlation Henry C. Caldwell, Paul N. Craig, and William G. Groves pp 1079 - 1081; DOI: 10.1021/jm00300a014 |
New s-triazine derivatives as depressants for reticuloendothelial hyperfunction induced by bacterial endotoxin Tsutomu Irikura, Yasuo Abe, Kyuya Okamura, Kyoichi Higo, Akitoshi Maeda, Fumihiko Morinaga, Goki Shirai, and Shinkichi Hatae pp 1081 - 1089; DOI: 10.1021/jm00300a015 |
Synthesis and pharmacological evaluation of .alpha.,.alpha.-disubstituted naphthylacetaldehydes Gianfranco Pala, Arturo Donetti, Antonio Mantegani, Elda Crescenzi, Bruno Lumachi, and Germano Coppi pp 1089 - 1092; DOI: 10.1021/jm00300a016 |
Synthesis and pharmacological properties of N-derivatives of 5,7,12,13-tetrahydro-6H-dibenz[c,g]azonine Silvano Casadio, Gianfranco Pala, Antonio Mantegani, Ernesta Marazzi-Uberti, Germano Coppi, and Carla Turba pp 1092 - 1095; DOI: 10.1021/jm00300a017 |
Specific competitive inhibition of L-asparaginyl transfer ribonucleic acid lygase by .beta.-aminoamides T. O. Yellin and M. R. Harnden pp 1095 - 1098; DOI: 10.1021/jm00300a018 |
Polypeptides. XLVII. Effect of the pyrazole-imidazole replacement on the biological activity of thyrotropin-releasing hormone Klaus Hofmann and Cyril Y. Bowers pp 1099 - 1101; DOI: 10.1021/jm00300a019 |
Antibacterial activity of nitrobenzofurans Larry J. Powers and Mathias P. Mertes pp 1102 - 1105; DOI: 10.1021/jm00300a020 |
Analogs of the antimalarial 2-bromo-N,N-bis(diethylaminoethyl)-4,5-dimethoxyaniline. 2-Position variations Eugene L. Stogryn pp 1106 - 1109; DOI: 10.1021/jm00300a021 |
Antimalarials. 1. Aminoalkylamino derivatives of 2,3-dihydrofuroquinolines Philip A Cruickshank, Fui Tseng Lee, and A. Lupichuk pp 1110 - 1114; DOI: 10.1021/jm00300a022 |
Chemistry of cephalosporin antibiotics. XX. Synthesis and biological properties of 3-acyloxymethyl-7-[2-(thienyl)acetamido]-3-cephem-4-carboxylic acid and related derivatives Stjepan Kukolja pp 1114 - 1117; DOI: 10.1021/jm00300a023 |
Carcinostatic activity of thiosemicarbazones of formyl heteroaromatic compounds. VI. 1-Formylisoquinoline derivatives bearing additional ring substituents, with notes on mechanism of action Frederic A. French, Erwin J. Blanz, Jefferson R. DoAmaral, and Douglas A. French pp 1117 - 1124; DOI: 10.1021/jm00300a024 |
Carcinostatic activity of thiosemicarbazones of formyl heteroaromatic compounds. VII. 2-Formylpyridine derivatives bearing additional ring substituents Frederic A. French, Erwin J. Blanz, Jefferson R. DoAmaral, and Douglas A. French pp 1124 - 1130; DOI: 10.1021/jm00300a025 |
Irreversible enzyme inhibitors. CLXXIII. Cure of Walker 256 ascites by reversible and irreversible inhibitors of dihydrofolic reductase derived from 1-(substituted-phenyl)-4,6-diamino-1,2-dihydro-2,2-dimethyl-s-triazine Bernard Randall Baker, Nicolaas M. J. Vermeulen, Wallace T. Ashton, and Adrian J. Ryan pp 1130 - 1140; DOI: 10.1021/jm00300a026 |
Irreversible enzyme inhibitors. CLXXIV. Metabolism of 4-[p-(4,6-diamino-1,2-dihydro-2,2-dimethyl-s-triazin-1-yl)hydrocinnamido]-o-toluenesulfonyl fluoride (NSC-113423), and active-site-directed irreversible inhibitor of dihydrofolic reductase Bernard Randall Baker, Adrian J. Ryan, and Nicolaas M. J. Vermeulen pp 1140 - 1142; DOI: 10.1021/jm00300a027 |
Irreversible enzyme inhibitors. CLXXV. Irreversible inhibition of purifed dihydrofolic reductase Bernard Randall Baker and Nicolaas M. J. Vermeulen pp 1143 - 1148; DOI: 10.1021/jm00300a028 |
Irreversible enzyme inhibitors. CLXXVI. Active-site-directed irreversible inhibitors of dihydrofolate reductase derived from 4,6-diamino-1,2-dihydro-2,2-dimethyl-1-phenyl-s-triazine by ether bridging to a terminal sulfonyl fluoride Bernard Randall Baker and Wallace T. Ashton pp 1149 - 1154; DOI: 10.1021/jm00300a029 |
Irreversible enzyme inhibitors. CLXXVII. Active-site-directed irreversible inhibitors of dihydrofolate reductase derived from 4,6-diamino-1,2-dihydro-2,2-dimethyl-1-(phenylalkylphenyl)-s-triazines. II Bernard Randall Baker and Nicolaas M. J. Vermeulen pp 1154 - 1160; DOI: 10.1021/jm00300a030 |
Irreversible enzyme inhibitors. CLXXVIII. Active-site-directed irreversible inhibitors of dihydrofolate reductase derived from 1-(4-benzyloxy-3-chlorophenyl)-4,6-diamino-1,2-dihydro-2,2-dimethyl-s-triazine with a terminal sulfonyl fluoride Bernard Randall Baker and Wallace T. Ashton pp 1161 - 1165; DOI: 10.1021/jm00300a031 |
Ireversible enzyme inhibitors. CLXXIX. Active-site-directed irreversible enzyme inhibitors of dihydrofolate reductase from 1-(3-chlorophenyl)-4,6-diamino-1,2-dihydro-2,2-dimethyl-s-triazine with oxyamide bridges to a terminal sulfonyl fluoride Bernard Randall Baker and Wallace T. Ashton pp 1165 - 1170; DOI: 10.1021/jm00300a032 |
Synthesis and biological activity of some 5-(1-adamantyl)pyrimidines. 1 James P. Jonak, Sigmund F. Zakrzewski, Lawrence H. Mead, and Maire T. Hakala pp 1170 - 1172; DOI: 10.1021/jm00300a033 |
Epoxide formation from (2S,3S)-threitol 1,4-bismethanesulfonate. Preparation and biological activity of (2S,3S)-1,2-epoxy-3,4-butanediol 4-methanesulfonate Peter W. Feit, Niels Rastrup-Andersen, and Rene Matagne pp 1173 - 1175; DOI: 10.1021/jm00300a034 |
Carbamate ester latentiation of physiologically active amines Leo G. Abood and Anthony J. Verbiscar pp 1176 - 1179; DOI: 10.1021/jm00300a035 |
Peripheral inhibition of thyroxine by thiohydantoins derived from amino acids Wilfred W. Westerfeld, Joseph V. Marx, and Dan A. Richert pp 1179 - 1181; DOI: 10.1021/jm00300a036 |
Molecular orbital study of 3,3'-5-trihalothyronine analogs Lemont B. Kier and James R. Hoyland pp 1182 - 1184; DOI: 10.1021/jm00300a037 |
Quantitative structure-activity models. Conditions for application and statistical interpretation William P. Purcell, Donna R. Hudson, and George E. Bass pp 1184 - 1189; DOI: 10.1021/jm00300a038 |
Structure-activity correlations for anticonvulsant drugs Eric J. C. Lien pp 1189 - 1191; DOI: 10.1021/jm00300a039 |
Parabolic relation between drug potency and hydrophobicity James W. McFarland pp 1192 - 1196; DOI: 10.1021/jm00300a040 |
Mass spectral analysis in the identification of human metabolites of warfarin William F. Trager, Richard J. Lewis, and William A. Garland pp 1196 - 1204; DOI: 10.1021/jm00300a041 |
Benzo[b]thiophene derivatives. XVI. Sulfur isosteres of melatonin, bufotenine, 5-hydroxytryptophan, and related structures Ernest Campaigne and Alan Dinner pp 1205 - 1208; DOI: 10.1021/jm00300a042 |
Isothiazolecarboxaldoximes and methylated derivatives as therapeutic agents in poisoning by organophosphorus compounds H. P. Benschop, A. M. Van Oosten, D. H. J. M. Platenburg, and C. Van Hooidonk pp 1208 - 1212; DOI: 10.1021/jm00300a043 |
Perfluoroalkyl carbonyl compounds. 1. Perfluoroaldehyde and perfluorocarboxylic acid derivatives Stephen S. Szinai, George Crank, and David R. K. Harding pp 1212 - 1215; DOI: 10.1021/jm00300a044 |
Perfluoroalkyl carbonyl compounds. 2. Derivatives of hexafluoroacetone Stephen S. Szinai, George Crank, and David R. K. Harding pp 1215 - 1217; DOI: 10.1021/jm00300a045 |
Structure-taste relation of aspartic acid amides Robert H. Mazur, Arthur H. Goldkamp, Patricia A. James, and James M. Schlatter pp 1217 - 1221; DOI: 10.1021/jm00300a046 |
12-Carboxyeudesma-3,11(13)-diene. Novel sesquiterpenic acid with a narrow antifungal spectrum Gad Shtacher and Yoel Kashman pp 1221 - 1223; DOI: 10.1021/jm00300a047 |
Acyl derivatives of 5-hydroxy-6,7-benzomorphans. Prodine congeners Mikio Takeda and Everette L. May pp 1223 - 1224; DOI: 10.1021/jm00300a048 |
Conformational study of .beta.-phenethanolamine receptor sites. IV. Synthesis of erythro- and threo-3-amino-2-phenyl-2-butanols Edward E. Smissman and Stanley J. Vickers pp 1224 - 1225; DOI: 10.1021/jm00300a049 |
2-Amino-5,6-dihydroxyindan-2-carboxylic acid. A potential hypotensive agent John William Lewis, John Bodenham Taylor, and Michael Jacklin pp 1226 - 1227; DOI: 10.1021/jm00300a050 |
Synthesis and pharmacology of a series of substituted 2-aminomethylpyrroles Stephen Raines and Csaba A. Kovacs pp 1227 - 1228; DOI: 10.1021/jm00300a051 |
New group of anorexigenic compounds Kurt Freter, Manfred Goetz, and James T. Oliver pp 1228 - 1230; DOI: 10.1021/jm00300a052 |
Tranquilizing drugs. Carbamates of 4-(4-hydroxypiperidino)-4'-fluorobutyrophenone and analogs Jorge P. Li, Robert G. Stein, John H. Biel, Jonas A. Gylys, and S. A. Ridlon pp 1230 - 1232; DOI: 10.1021/jm00300a053 |
Biphenylene derivatives with pharmacophoric side chains Alfred Burger and Sharon S. Hillery pp 1232 - 1233; DOI: 10.1021/jm00300a054 |
Synthesis of potential antimalarial agents. VI. Preparation of 3-(p-chlorophenyl)-8-{[4-(diethylamino)-1-methylbutyl]amino}pyrido[2,3-b]pyrazine Carroll Temple, Jerry D. Rose, and John A. Montgomery pp 1234 - 1235; DOI: 10.1021/jm00300a055 |
Hydroxylamine derivatives as potential antimalarial agents. 1. Hydroxamic acids John B. Hynes pp 1235 - 1237; DOI: 10.1021/jm00300a056 |
Organic fluorine compounds. IV. Synthesis and antifungal properties of 2-fluoro fatty acid amides Herman Gershon, Raymond L. Rodin, Raulo Parmegiani, and Patricia K. Godfrey pp 1237 - 1239; DOI: 10.1021/jm00300a057 |
Analogs of 1-(4-dimethylaminobenzylidene)indene. Modifications of the amino group Carl T. Bahner, David H. Brotherton, Mary K. Brotherton, Harry Harmon, Norma H. Bingham, Lydia M. Rivers, and Stuart L. Watson pp 1240 - 1242; DOI: 10.1021/jm00300a058 |
5'-Diazogriseofulvin Howard Newman, Thomas L. Fields, and Robert B. Angier pp 1242 - 1243; DOI: 10.1021/jm00300a059 |
Steroids and related natural products. 63. 17.beta.-Acetoxy-4-oxa-2-androstene George R. Pettit and Tirumalai R. Kasturi pp 1244 - 1245; DOI: 10.1021/jm00300a060 |
Hypocholesteremic agents. 2. Cyclohexane and indan derivatives Frank J. Villani and Claire A. Ellis pp 1245 - 1246; DOI: 10.1021/jm00300a061 |
1-Dodecylpyridinium dodecyl sulfate Gunther S Fonken and Forrest A. MacKellar pp 1246 - 1246; DOI: 10.1021/jm00300a062 |
SH analog of the estrogen hexestrol Lars Terenius pp 1246 - 1247; DOI: 10.1021/jm00300a063 |
Compounds related to insect juvenile hormone. V. Derivatives of citronellol and citronellylamine Philip E. Sonnet, Meyer Schwarz, and Nobel Wakabayashi pp 1247 - 1248; DOI: 10.1021/jm00300a064 |
Synthesis of new urethans. p-Ethylsulfonyl- and p-dimethylsulfamoylcarbanilic acid esters N. Sharghi, Iradj Lalezari, Gh. Niloofari, and F. Ghabgharan pp 1248 - 1248; DOI: 10.1021/jm00300a065 |
Synthesis of 5,7-dimethoxyindole P. J. Mulligan and S. La Berge pp 1248 - 1249; DOI: 10.1021/jm00300a066 |
Dithienylpiperidylthenilates Robert D. Schuetz and George P. Nilles pp 1249 - 1249; DOI: 10.1021/jm00300a067 |
Acetylenics. 1. Aromatic amines containing the acetylenic triple bond David Z. Simon, Romano L. Salvador, and Gaston Champagne pp 1249 - 1250; DOI: 10.1021/jm00300a068 |
Antifungal activity and geometric isomerism. Anilides of o-coumaric acid Alex Gringauz pp 1250 - 1250; DOI: 10.1021/jm00300a069 |
Potential antidiabetics. VI. 3-Methyl-4-arylhydrazono-2-isoxazolin-5-ones and 3-methyl-4-arylazo-5-(methyl phenyl)isoxazoles Hari G. Garg and Prem Pal Singh pp 1250 - 1251; DOI: 10.1021/jm00300a070 |
Pyrolysis of 1-adamantyl azidomethyl ketone Leo H. Sternbach and Robert Y. Ning pp 1251 - 1252; DOI: 10.1021/jm00300a071 |
Book Reviews pp 1252 - 1253; DOI: 10.1021/jm00300a600 |
Additions and Corrections - β-Adrenergic Blocking Agents. V. 1-Amino-3-(substituted phenoxy)-2-propanols. A. F. Crowther, D. J. Gilman, B. J .McLoughlin, L. H. Smith, R. W. Turner, and T. M. Wood pp 1253 - 1253; DOI: 10.1021/jm00300a601 |
Additions and Corrections - Hypotensive Agents. (+)- and (-)-2-Methoxy-2-(3-methoxyphenyl)ethyl-amine and Related Compounds. R. Howe, E. H .P. Young, and A. D. Ainley pp 1253 - 1253; DOI: 10.1021/jm00300a602 |
Additions and Corrections - Irreversible Enzyme Inhibitors. CLXVIII. B. R .Baker, N. M. Vermeulen, and A. J .Ryan pp 1253 - 1253; DOI: 10.1021/jm00300a603 |
Additions and Corrections - Coumarin Derivatives as Coronary Vasodilators. D. S. Bariana pp 1253 - 1253; DOI: 10.1021/jm00300a604 |